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Carbamazepine

Anticonvulsant • Last reviewed 2025-09-24

Brands: Tegretol

Sources updated 20251 references

Summary

General Information

Anticonvulsant

Dosage & Administration

Typical dose range: 400–1200 mg/day (in divided doses)

Therapeutic level: 4000–12000 ng/mL

Indications (label)

Mechanism (brief)

Voltage‑gated sodium channel blocker; reduces high‑frequency neuronal firing.

Metabolism & Half‑life

  • Metabolism: Strong CYP3A4 inducer; autoinduction; epoxide metabolite.
  • Half‑life: ~12–17 h (after autoinduction).

Therapeutic Drug Monitoring (TDM)

Recommended: Yes

Reference range: 400012000 ng/mL

Sampling: Trough

Source: AGNP 2018

References