Oxcarbazepine
Anticonvulsant • Last reviewed 2025-09-26
Brands: Trileptal, Oxtellar XR
Sources updated 2025 • 1 references
General Information
Indicated for: Seizures (partial-onset); sometimes used off-label as adjunctive mood stabilizer. Anticonvulsant
Dosage & Administration
Typical dose range: 900–1500 mg/day (divided or XR)
Indications (label)
Seizures (partial-onset); sometimes used off-label as adjunctive mood stabilizer.
View labelExact
Mechanism (brief)
Voltage-gated sodium channel modulator reducing glutamate release.
Metabolism & Half‑life
- Metabolism: Cytosolic reduction to active MHD; induces CYP3A4 and UGT.
- Half‑life: ~9 h (MHD).
Therapeutic Drug Monitoring (TDM)
Recommended: No
References
- Oxcarbazepine labelExact (2025)